Allosteric Inhibitor TREA-0236 Containing Non-hydrolysable Quinazoline-4-one for EGFR T790M/C797S Mutants Inhibition

Seoyoung Lee, Jiwon Kim, Krishna Babu Duggirala, Areum Go, Inji Shin, Byoung Chul Cho, Gildon Choi, Chong Hak Chae, Kwangho Lee

Research output: Contribution to journalArticlepeer-review

20 Scopus citations
Original languageEnglish
Pages (from-to)895-898
Number of pages4
JournalBulletin of the Korean Chemical Society
Volume39
Issue number7
DOIs
StatePublished - Jul 2018

Keywords

  • Allosteric inhibitor
  • EAI045
  • EGFR T790M/C797S
  • Kinases
  • NSCLC

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